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Design, Synthesis, and Biological Evaluation of Novel Thioureidobenzamide (TBA) Derivatives as HBV Capsid Assembly Modulators.

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第一作者: Mei,Wang
第一单位: School of Pharmacy, Weifang Medical University, Weifang 261053, Shandong, P. R. China.
作者: Mei,Wang [1] ; Jian,Zhang [1] ; Yutong,Dou [2] ; Minghui,Liang [1] ; Yong,Xie [3] ; Peng,Xue [4] ; Linyue,Liu [1] ; Chuanju,Li [5] ; Yuanze,Wang [6] ; Feiyan,Tao [4] ; Xiaohui,Zhang [7] ; Huili,Hu [7] ; Kairui,Feng [1] ; Lei,Zhang [1] ; Zhuanchang,Wu [2] ; Yunfu,Chen [3] ; Peng,Zhan [8] ; Haiyong,Jia [1]
作者单位: School of Pharmacy, Weifang Medical University, Weifang 261053, Shandong, P. R. China. [1] Key Laboratory for Experimental Teratology of Ministry of Education, Key Laboratory of Infection and Immunity of Shandong Province and Dept. Immunology, School of Basic Medical Sciences, Qilu Hospital, Cheeloo Medical College, Shandong University, Jinan 250012, Shandong, P. R. China. [2] State Key Laboratory of Anti-Infective Drug Development (NO. 2015DQ780357), Sunshine Lake Pharma Co., Ltd, Dongguan 523871, P. R. China. [3] School of Public Health, Weifang Medical University, Weifang 261053, Shandong, P. R. China. [4] Department of Pharmacy, Affiliated Hospital of Jining Medical University, Jining 272000, Shandong, P. R. China. [5] Guangzhou Laboratory, Guangzhou International Bio Island, Guangzhou 510000, Guangdong, P. R. China. [6] Key Laboratory of Experimental Teratology, Ministry of Education and Department of Genetics, School of Basic Medical Sciences, Qilu Hospital, Cheeloo Medical College, Shandong University, Jinan 250012, P. R. China.;The Research Center of Stem Cell and Regenerative Medicine, Department of Systems Biomedicine, School of Basic Medical Sciences, Cheeloo College of Medicine, Shandong University, Jinan 250012, P. R. China. [7] Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Shandong University, 44 West Culture Road, 250012 Jinan, Shandong, P. R. China. [8]
DOI 10.1021/acs.jmedchem.3c01022
PMID 37839070
发布时间 2023-10-27
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Journal of medicinal chemistry

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