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Uncovering PROTAC Sensitivity and Efficacy by Multidimensional Proteome Profiling: A Case for STAT3.

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第一作者: Yuying,Suo
第一单位: University of Chinese Academy of Sciences, NO.19A Yuquan Road, Beijing 100049, P. R. China.;Department of Analytical Chemistry, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica Chinese Academy of Sciences, Shanghai 201203, China.
作者: Yuying,Suo [1] ; Daohai,Du [2] ; Chao,Chen [3] ; Hongwen,Zhu [4] ; Xiongjun,Wang [5] ; Nixue,Song [4] ; Dayun,Lu [4] ; Yaxi,Yang [6] ; Jiacheng,Li [2] ; Jun,Wang [2] ; Zhongyuan,Luo [2] ; Bing,Zhou [6] ; Cheng,Luo [7] ; Hu,Zhou [8]
作者单位: University of Chinese Academy of Sciences, NO.19A Yuquan Road, Beijing 100049, P. R. China.;Department of Analytical Chemistry, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica Chinese Academy of Sciences, Shanghai 201203, China. [1] Drug Discovery and Design Center, the Center for Chemical Biology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China. [2] Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai 201203, China.;Shandong Laboratory of Yantai Drug Discovery, Bohai Rim Advanced Research Institute for Drug Discovery, Yantai, Shandong 264117, China.;State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China. [3] Department of Analytical Chemistry, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica Chinese Academy of Sciences, Shanghai 201203, China. [4] Precise Genome Engineering Center, School of Life Sciences, Guangzhou University, Guangzhou 510006, China. [5] University of Chinese Academy of Sciences, NO.19A Yuquan Road, Beijing 100049, P. R. China.;School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, University of Chinese Academy of Sciences, Hangzhou 310024, China.;Shandong Laboratory of Yantai Drug Discovery, Bohai Rim Advanced Research Institute for Drug Discovery, Yantai, Shandong 264117, China.;State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China. [6] School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, University of Chinese Academy of Sciences, Hangzhou 310024, China.;Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Zhongshan 528437, China.;Drug Discovery and Design Center, the Center for Chemical Biology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China. [7] University of Chinese Academy of Sciences, NO.19A Yuquan Road, Beijing 100049, P. R. China.;School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, University of Chinese Academy of Sciences, Hangzhou 310024, China.;Department of Analytical Chemistry, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica Chinese Academy of Sciences, Shanghai 201203, China. [8]
DOI 10.1021/acs.jmedchem.3c02371
PMID 38466231
发布时间 2025-01-29
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Journal of medicinal chemistry

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