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DrugMap: A quantitative pan-cancer analysis of cysteine ligandability.

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作者: Mariko,Takahashi [1] ; Harrison B,Chong [2] ; Siwen,Zhang [2] ; Tzu-Yi,Yang [2] ; Matthew J,Lazarov [2] ; Stefan,Harry [3] ; Michelle,Maynard [4] ; Brendan,Hilbert [4] ; Ryan D,White [4] ; Heather E,Murrey [4] ; Chih-Chiang,Tsou [4] ; Kira,Vordermark [2] ; Jonathan,Assaad [2] ; Magdy,Gohar [2] ; Benedikt R,Dürr [2] ; Marianne,Richter [2] ; Himani,Patel [2] ; Gregory,Kryukov [4] ; Natasja,Brooijmans [4] ; Aliyu Sidi Omar,Alghali [5] ; Karla,Rubio [5] ; Antonio,Villanueva [5] ; Junbing,Zhang [2] ; Maolin,Ge [2] ; Farah,Makram [2] ; Hanna,Griesshaber [2] ; Drew,Harrison [2] ; Ann-Sophie,Koglin [2] ; Samuel,Ojeda [2] ; Barbara,Karakyriakou [2] ; Alexander,Healy [2] ; George,Popoola [2] ; Inbal,Rachmin [6] ; Neha,Khandelwal [2] ; Jason R,Neil [4] ; Pei-Chieh,Tien [2] ; Nicholas,Chen [7] ; Tobias,Hosp [2] ; Sanne,van den Ouweland [2] ; Toshiro,Hara [5] ; Lillian,Bussema [5] ; Rui,Dong [5] ; Lei,Shi [2] ; Martin Q,Rasmussen [2] ; Ana Carolina,Domingues [2] ; Aleigha,Lawless [8] ; Jacy,Fang [9] ; Satoshi,Yoda [2] ; Linh Phuong,Nguyen [2] ; Sarah Marie,Reeves [2] ; Farrah Nicole,Wakefield [2] ; Adam,Acker [2] ; Sarah Elizabeth,Clark [2] ; Taronish,Dubash [2] ; John,Kastanos [2] ; Eugene,Oh [10] ; David E,Fisher [6] ; Shyamala,Maheswaran [10] ; Daniel A,Haber [11] ; Genevieve M,Boland [12] ; Moshe,Sade-Feldman [10] ; Russell W,Jenkins [13] ; Aaron N,Hata [10] ; Nabeel M,Bardeesy [10] ; Mario L,Suvà [14] ; Brent R,Martin [4] ; Brian B,Liau [15] ; Christopher J,Ott [10] ; Miguel N,Rivera [14] ; Michael S,Lawrence [16] ; Liron,Bar-Peled [17]
作者单位: Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA. Electronic address: mtaka@umich.edu. [1] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA. [2] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Department of Chemistry and Chemical Biology, Harvard University, Cambridge, MA 02138, USA. [3] Scorpion Therapeutics, Boston, MA 02110, USA. [4] Department of Pathology, Massachusetts General Hospital, Boston, MA 02114, USA. [5] Cutaneous Biology Research Center, Massachusetts General Hospital, Boston, MA 02114, USA. [6] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Department of Pathology, Harvard Medical School, Boston, MA 02114, USA. [7] Department of Surgery, Massachusetts General Hospital, Boston, MA 02114, USA; Broad Institute of MIT and Harvard, Cambridge, MA 02142, USA. [8] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Broad Institute of MIT and Harvard, Cambridge, MA 02142, USA. [9] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Department of Medicine, Harvard Medical School, Boston, MA 02114, USA. [10] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Department of Medicine, Harvard Medical School, Boston, MA 02114, USA; Howard Hughes Medical Institute, Chevy Chase, MD 20815, USA. [11] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Department of Surgery, Massachusetts General Hospital, Boston, MA 02114, USA; Broad Institute of MIT and Harvard, Cambridge, MA 02142, USA; Department of Surgery, Harvard Medical School, Boston, MA 02114, USA. [12] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Broad Institute of MIT and Harvard, Cambridge, MA 02142, USA; Department of Medicine, Harvard Medical School, Boston, MA 02114, USA. [13] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Department of Pathology, Massachusetts General Hospital, Boston, MA 02114, USA; Broad Institute of MIT and Harvard, Cambridge, MA 02142, USA; Department of Pathology, Harvard Medical School, Boston, MA 02114, USA. [14] Department of Chemistry and Chemical Biology, Harvard University, Cambridge, MA 02138, USA. [15] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Broad Institute of MIT and Harvard, Cambridge, MA 02142, USA; Department of Pathology, Harvard Medical School, Boston, MA 02114, USA. Electronic address: mslawrence@mgh.harvard.edu. [16] Krantz Family Center for Cancer Research, Massachusetts General Hospital Cancer Center, Charlestown, MA 02129, USA; Department of Medicine, Harvard Medical School, Boston, MA 02114, USA. Electronic address: lbar-peled@mgh.harvard.edu. [17]
DOI 10.1016/j.cell.2024.03.027
PMID 38653237
发布时间 2025-02-05
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Cell

Cell

2024年187卷10期

2536-2556.e30页

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