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Kinetics of the inhibition of CYP3A4 and CYP2C19 activity by jabara juice and identification of the responsible inhibitory components.

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作者单位: Division of Clinical Pharmacy, Graduate School of Pharmaceutical Sciences, Keio University, 1-5-30 Shibakoen, Minato-ku, Tokyo, 105-8512, Japan. [1] Division of Clinical Pharmacy Faculty of Pharmacy, Keio University, 1-5-30 Shibakoen, Minato-ku, Tokyo, 105-8512, Japan. [2] Division of Drugs, National Institute of Health Sciences, 3-25-26 Tonomachi, Kawasaki-ku, Kawasaki City, Kanagawa, 210-9501, Japan. [3] Division of Natural Medicines, Faculty of Pharmacy, Keio University, 1-5-30 Shibakoen, Minato-ku, Tokyo, 105-8512, Japan. [4] Department of Pharmacy, University of Ryukyus Hospital, 207 Uehara, Nishihara-cho, Okinawa, 903-0215, Japan. [5] Laboratory of Drug Metabolism and Pharmacokinetics, Showa Pharmaceutical University, 3-2-1 Higashi-Tamagawagakuen, Machidashi, Tokyo, 194-8543, Japan. [6] Department of Biochemistry, Vanderbilt University School of Medicine, 2200 Pierce Avenue, Nashville, TN 37232, United States. [7] Gunma University Graduate School of Medicine, 3-39-22 Showa-machi, Maebashi City, Gunma, 371-8511, Japan. [8] Division of Clinical Pharmacy Faculty of Pharmacy, Keio University, 1-5-30 Shibakoen, Minato-ku, Tokyo, 105-8512, Japan; Department of Clinical Pharmacy, Keio University School of Medicine, 35 Shinanomachi, Shinjuku-ku, Tokyo, 160-8582, Japan. [9] Division of Clinical Pharmacy, Graduate School of Pharmaceutical Sciences, Keio University, 1-5-30 Shibakoen, Minato-ku, Tokyo, 105-8512, Japan; Division of Clinical Pharmacy Faculty of Pharmacy, Keio University, 1-5-30 Shibakoen, Minato-ku, Tokyo, 105-8512, Japan; Department of Clinical Pharmacy, Keio University School of Medicine, 35 Shinanomachi, Shinjuku-ku, Tokyo, 160-8582, Japan. [10] Division of Clinical Pharmacy, Graduate School of Pharmaceutical Sciences, Keio University, 1-5-30 Shibakoen, Minato-ku, Tokyo, 105-8512, Japan; Division of Clinical Pharmacy Faculty of Pharmacy, Keio University, 1-5-30 Shibakoen, Minato-ku, Tokyo, 105-8512, Japan; Department of Clinical Pharmacy, Keio University School of Medicine, 35 Shinanomachi, Shinjuku-ku, Tokyo, 160-8582, Japan; Department of Pharmacy, Keio University Hospital, 35 Shinanomachi, Shinjuku-ku, Tokyo, 160-8582, Japan. Electronic address: ohtani@keio.jp. [11]
DOI 10.1016/j.xphs.2024.10.037
PMID 39481475
发布时间 2024-11-21
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