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A Target Class Ligandability Evaluation of WD40 Repeat-Containing Proteins.

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作者: Suzanne,Ackloo [1] ; Fengling,Li [1] ; Magda,Szewczyk [1] ; Almagul,Seitova [1] ; Peter,Loppnau [1] ; Hong,Zeng [1] ; Jin,Xu [2] ; Shabbir,Ahmad [1] ; Yelena A,Arnautova [3] ; A J,Baghaie [3] ; Serap,Beldar [1] ; Albina,Bolotokova [1] ; Paolo A,Centrella [4] ; Irene,Chau [1] ; Matthew A,Clark [4] ; John W,Cuozzo [5] ; Saba,Dehghani-Tafti [1] ; Jeremy S,Disch [5] ; Aiping,Dong [1] ; Antoine,Dumas [3] ; Jianwen A,Feng [2] ; Pegah,Ghiabi [1] ; Elisa,Gibson [1] ; Justin,Gilmer [2] ; Brian,Goldman [5] ; Stuart R,Green [1] ; Marie-Aude,Guié [4] ; John P,Guilinger [4] ; Nathan,Harms [3] ; Oleksandra,Herasymenko [1] ; Scott,Houliston [6] ; Ashley,Hutchinson [1] ; Steven,Kearnes [7] ; Anthony D,Keefe [4] ; Serah W,Kimani [1] ; Trevor,Kramer [5] ; Maria,Kutera [1] ; Haejin A,Kwak [1] ; Cristina,Lento [8] ; Yanjun,Li [1] ; Jenny,Liu [4] ; Joachim,Loup [9] ; Raquel A C,Machado [1] ; Christopher J,Mulhern [10] ; Sumera,Perveen [1] ; Germanna L,Righetto [1] ; Patrick,Riley [7] ; Suman,Shrestha [1] ; Eric A,Sigel [3] ; Madhushika,Silva [1] ; Michael D,Sintchak [11] ; Belinda L,Slakman [12] ; Rhys D,Taylor [4] ; James,Thompson [2] ; Wen,Torng [2] ; Carl,Underkoffler [5] ; Moritz,von Rechenberg [5] ; Ryan T,Walsh [4] ; Ian,Watson [2] ; Derek J,Wilson [8] ; Esther,Wolf [8] ; Manisha,Yadav [1] ; Aliakbar K,Yazdi [1] ; Junyi,Zhang [5] ; Ying,Zhang [4] ; Vijayaratnam,Santhakumar [1] ; Aled M,Edwards [1] ; Dalia,Barsyte-Lovejoy [13] ; Matthieu,Schapira [13] ; Peter J,Brown [1] ; Levon,Halabelian [13] ; Cheryl H,Arrowsmith [14]
作者单位: Structural Genomics Consortium, University of Toronto, 101 College St., Toronto, ON M5G 1L7, Canada. [1] Google, 1600 Amphitheatre Parkway, Mountain View, California 94043, United States. [2] ZebiAI Inc., 100 Beaver St., Waltham, Massachusetts 02435, United States. [3] X-Chem Inc., 100 Beaver St., Waltham, Massachusetts 02435, United States. [4] ZebiAI Inc., 100 Beaver St., Waltham, Massachusetts 02435, United States.;Relay Therapeutics, 399 Binney St., Cambridge, Massachusetts 02139, United States. [5] Princess Margaret Cancer Centre, University of Toronto, Toronto, ON M5G 2M9, Canada. [6] Google, 1600 Amphitheatre Parkway, Mountain View, California 94043, United States.;Relay Therapeutics, 399 Binney St., Cambridge, Massachusetts 02139, United States. [7] Department of Chemistry, York University, Toronto, ON M3J 1P3, Canada. [8] Department of Chemistry, University of Toronto, Toronto, ON M5S 3H6, Canada. [9] ZebiAI Inc., 100 Beaver St., Waltham, Massachusetts 02435, United States.;X-Chem Inc., 100 Beaver St., Waltham, Massachusetts 02435, United States. [10] Civetta Therapeutics, 10 Wilson Rd., Cambridge, Massachusetts 02138, United States. [11] ZebiAI Inc., 100 Beaver St., Waltham, Massachusetts 02435, United States.;X-Chem Inc., 100 Beaver St., Waltham, Massachusetts 02435, United States.;Relay Therapeutics, 399 Binney St., Cambridge, Massachusetts 02139, United States. [12] Structural Genomics Consortium, University of Toronto, 101 College St., Toronto, ON M5G 1L7, Canada.;Department of Pharmacology and Toxicology, University of Toronto, Toronto, ON M5S 1A8, Canada. [13] Structural Genomics Consortium, University of Toronto, 101 College St., Toronto, ON M5G 1L7, Canada.;Princess Margaret Cancer Centre, University of Toronto, Toronto, ON M5G 2M9, Canada. [14]
DOI 10.1021/acs.jmedchem.4c02010
PMID 39495097
发布时间 2025-01-23
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Journal of medicinal chemistry

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