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Development of Oral, Potent, and Selective CK1α Degraders for AML Therapy.

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作者: Lu,Huang [1] ; Lu,Chen [2] ; Lu,Chen [3] ; Bo,Peng [3] ; Lixin,Zhou [4] ; Yanli,Sun [3] ; Taiting,Shi [5] ; Jiayi,Lu [6] ; Weiye,Lin [7] ; Yuhang,Liu [8] ; Linhui,Cao [8] ; Lanlan,Li [9] ; Qiangqiang,Han [10] ; Xi,Chen [10] ; Ping,Yang [11] ; Shuo,Zhang [11] ; Zhe,Wang [11] ; Jing,Yang [4] ; Zhixiang,Guo [11] ; Baishan,Jiang [2] ; Wenchao,Lu [3]
作者单位: Department of Cardiovascular Surgery, The First Affiliated Hospital of Anhui Medical University, 218 Jixi Road, Hefei 230022, China.;Lingang Laboratory, Shanghai 200031, China. [1] Department of Radiation and Medical Oncology, Medical Research Institute, Frontier Science Center of Immunology and Metabolism, Zhongnan Hospital of Wuhan University, School of Pharmaceutical Sciences, Wuhan University, Wuhan 430071, China. [2] Lingang Laboratory, Shanghai 200031, China. [3] Department of Hematology, Tongji Hospital, Frontier Science Center for Stem Cell Research, Shanghai Key Laboratory of Signaling and Disease Research, School of Life Sciences and Technology, Tongji University, Shanghai 200092, China. [4] Lingang Laboratory, Shanghai 200031, China.;Department of Neurosurgery, The First Affiliated Hospital of Wenzhou Medical University, Wenzhou 325000, China. [5] College of Science, Northeastern University, 360 Huntington Avenue, Boston, Massachusetts 02115, United States. [6] Lingang Laboratory, Shanghai 200031, China.;School of Life Science and Technology, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai 201210, China. [7] Lingang Laboratory, Shanghai 200031, China.;School of Pharmacy, Key Laboratory of Molecular Pharmacology and Drug Evaluation (Yantai University), Ministry of Education; Collaborative Innovation Center of Advanced Drug Delivery System and Biotech Drugs in Universities of Shandong, Yantai University, Yantai 264005, China. [8] Lingang Laboratory, Shanghai 200031, China.;Institute of Entomology, The Provincial Special Key Laboratory for Development and Utilization of Insect Resources, Guizhou University, Guiyang 550025, China. [9] SpecAlly Life Technology Co., Ltd., Wuhan 430075, China. [10] Department of Cardiovascular Surgery, The First Affiliated Hospital of Anhui Medical University, 218 Jixi Road, Hefei 230022, China. [11]
DOI 10.1021/jacsau.4c00762
PMID 39610741
发布时间 2024-11-30
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JACS Au

JACS Au

2024年4卷11期

4423-4434页

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