Discovery of pyridine-based derivatives as FLT3 inhibitors for the treatment of acute myeloid leukemia.
作者:
主题词
动物(Animals);人类(Humans);小鼠(Mice);大鼠(Rats);抗肿瘤药(Antineoplastic Agents);细胞凋亡(Apoptosis);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物发现(Drug Discovery);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);fms样酪氨酸激酶3(fms-Like Tyrosine Kinase 3);白血病, 髓样, 急性(Leukemia, Myeloid, Acute);分子结构(Molecular Structure);蛋白激酶抑制剂(Protein Kinase Inhibitors);吡啶类(Pyridines);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);构效关系(Structure-Activity Relationship);三唑类(Triazoles)
DOI
10.1016/j.ejmech.2024.117173
PMID
39705732
发布时间
2025-01-03
- 浏览1
相似文献
- 中文期刊
- 外文期刊
- 学位论文
- 会议论文