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Discovery of pyridine-based derivatives as FLT3 inhibitors for the treatment of acute myeloid leukemia.

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作者: Beijing,Chen [1] ; Zhongyuan,Wang [2] ; Qi,Chen [2] ; Ying,Zhang [1] ; Shengfei,Wu [1] ; Yu,Zhang [1] ; Aihong,Li [1] ; Weiwei,Ouyang [3] ; Lijie,Sima [4] ; Xiaoxu,Li [3] ; Dongsheng,Zhao [1] ; Bilan,Luo [5] ; Jianta,Wang [1] ; Lei,Tang [6] ; Xiaoming,Su [7] ; Weike,Liao [8]
作者单位: Guizhou Provincial Engineering Technology Research Center for Chemical Drug R&D, Guizhou Medical University, Guiyang, 550004, China. [1] Department of Pharmacy, Guizhou Provincial People's Hospital, Guiyang, 550002, China. [2] Department of Oncology, The Affiliated Hospital of Guizhou Medical University and Cancer Hospital of Guizhou Medical University, Guiyang, 550001, China. [3] Department of Radiation Oncology, The Ninth Medical Center of Chinese PLA General Hospital, Beijing, 100101, China. [4] Advanced Innovation Center for Human Brain Protection, National Clinical Research Center for Geriatric Disorders, Xuanwu Hospital, Capital Medical University, Beijing, 100053, China. [5] Guizhou Provincial Engineering Technology Research Center for Chemical Drug R&D, Guizhou Medical University, Guiyang, 550004, China. Electronic address: tlei1974@gmc.edu.cn. [6] Department of Radiation Oncology, The Ninth Medical Center of Chinese PLA General Hospital, Beijing, 100101, China. Electronic address: smallcatsxm2022@163.com. [7] Guizhou Provincial Engineering Technology Research Center for Chemical Drug R&D, Guizhou Medical University, Guiyang, 550004, China. Electronic address: liaoweike2009@126.com. [8]
DOI 10.1016/j.ejmech.2024.117173
PMID 39705732
发布时间 2025-01-03
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