Repurposing the Antihypertensive Agent Hydralazine As an Inhibitor of the Base Excision Repair Enzyme APE1.
第一作者:
Tanhaul,Islam
第一单位:
University of Missouri, Department of Chemistry, 125 Chemistry Building, Columbia, Missouri 65211, United States.
作者:
主题词
肼苯哒嗪(Hydralazine);DNA-(无嘌呤或无嘧啶位点)裂合酶(DNA-(Apurinic or Apyrimidinic Site) Lyase);人类(Humans);抗高血压药(Antihypertensive Agents);DNA修复(DNA Repair);药物重新定位(Drug Repositioning);酶抑制剂(Enzyme Inhibitors);细胞系, 肿瘤(Cell Line, Tumor);抗肿瘤药(Antineoplastic Agents);分子结构(Molecular Structure);羟胺类(Hydroxylamines)
DOI
10.1021/acs.chemrestox.4c00445
PMID
39718352
发布时间
2025-01-20
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