A calmodulin-derived peptide TI-16 inhibits Alzheimer's disease progression by decreasing -Aβ burden and restoring calcium dyshomeostasis.
第一作者:
Jingyang,Su
第一单位:
Department of Pharmaceutical Toxicology, School of Pharmacy, China Medical University, Shenyang 110122, China; Department of Clinical Pharmacology, School of Pharmacy, China Medical University, Shenyang 110122, China.
作者:
医学主题词
阿尔茨海默病(Alzheimer Disease);钙(Calcium);动物(Animals);淀粉样β肽类(Amyloid beta-Peptides);钙调蛋白(Calmodulin);人类(Humans);小鼠(Mice);内环境稳定(Homeostasis);肽类(Peptides);细胞凋亡(Apoptosis);肽碎片(Peptide Fragments);剂量效应关系, 药物(Dose-Response Relationship, Drug);男(雄)性(Male);构效关系(Structure-Activity Relationship);分子结构(Molecular Structure);神经保护药(Neuroprotective Agents);疾病恶化(Disease Progression)
DOI
10.1016/j.bioorg.2025.108502
PMID
40280012
发布时间
2026-04-21
- 浏览0
Bioorganic chemistry
108502页
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