An adamantylureido-benzylamide aniline as FLAP/sEH dual inhibitor: Rational design, in vitro and in vivo lipidomic profiling.
第一作者:
Tania,Ciaglia
第一单位:
Department of Pharmacy, University of Salerno, Via G. Paolo II 132, Fisciano, Salerno, Italy, 84084.
作者:
医学主题词
环氧水解酶类(Epoxide Hydrolases);苯胺化合物(Aniline Compounds);人类(Humans);药物设计(Drug Design);动物(Animals);5-脂氧合酶活化蛋白类(5-Lipoxygenase-Activating Proteins);分子结构(Molecular Structure);构效关系(Structure-Activity Relationship);5-脂氧合酶活化蛋白抑制剂(5-Lipoxygenase-Activating Protein Inhibitors);酶抑制剂(Enzyme Inhibitors);金刚烷(Adamantane);剂量效应关系, 药物(Dose-Response Relationship, Drug);男(雄)性(Male)
DOI
10.1016/j.ejmech.2025.118338
PMID
41197472
发布时间
2025-12-03
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