Discovery of γ-Tetrahydrocarboline Derivatives as <i>Plasmodium falciparum</i> Histone Deacetylase Inhibitors for Treatment of Malaria.
第一作者:
Hao,Ni
第一单位:
Institute of Drug Discovery and Design, College of Pharmaceutical Sciences, Zhejiang University, Hangzhou 310058, China.
作者:
医学主题词
恶性疟原虫(Plasmodium falciparum);抗疟药(Antimalarials);人类(Humans);组蛋白脱乙酰基酶抑制剂(Histone Deacetylase Inhibitors);咔啉类(Carbolines);动物(Animals);构效关系(Structure-Activity Relationship);药物发现(Drug Discovery);疟疾(Malaria);疟疾, 恶性(Malaria, Falciparum);小鼠(Mice);组蛋白脱乙酰基酶1(Histone Deacetylase 1)
DOI
10.1021/acs.jmedchem.5c02869
PMID
41485139
发布时间
2026-01-22
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Journal of medicinal chemistry
1434-1453页
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