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Identification of an N-methylpyrazole derivative as a selective inhibitor of breast cancer resistance protein (BCRP/ABCG2).

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第一单位: Graduate Program in Pharmaceutical Sciences, Laboratory of Cancer Drug Resistance, Federal University of Parana, Curitiba, 80210-170, PR, Brazil.
作者单位: Graduate Program in Pharmaceutical Sciences, Laboratory of Cancer Drug Resistance, Federal University of Parana, Curitiba, 80210-170, PR, Brazil. [1] Graduate Program in Pharmaceutical Sciences, Laboratory of Cancer Drug Resistance, Federal University of Parana, Curitiba, 80210-170, PR, Brazil; Interfaculty Institute of Microbiology and Infection Medicine (IMIT), DZIF Tübingen Partner Site. University Hospital Tübingen, Tübingen, Germany. [2] Laboratory for Synthesis of Heterocycles (SINTHET), Chemistry Department, State University of Maringá- UEM, Maringá, Paraná 87020-900, Brazil. [3] Interfaculty Institute of Microbiology and Infection Medicine (IMIT), DZIF Tübingen Partner Site. University Hospital Tübingen, Tübingen, Germany; School of Pharmacy, Faculty of Health Sciences, University of Eastern Finland, P.O. Box 1627, FI-70211 Kuopio, Finland. [4] Graduate Program in Pharmaceutical Sciences, Federal University of Parana, Curitiba, 80210-170, PR, Brazil. [5] Gastroenterology and Technologies for Health Team, Centre de Recherche en Cancérologie de Lyon, Centre Léon Bérard, CNRS 5286, INSERM 1052, Université Claude Bernard Lyon 1, Univ Lyon, 69373, Lyon, France. [6] Université Grenoble Alpes, INSERM, LRB, 38000, Grenoble, France. [7] Graduate Program in Pharmaceutical Sciences, Laboratory of Cancer Drug Resistance, Federal University of Parana, Curitiba, 80210-170, PR, Brazil. Electronic address: gvaldameri@ufpr.br. [8] Graduate Program in Pharmaceutical Sciences, Laboratory of Cancer Drug Resistance, Federal University of Parana, Curitiba, 80210-170, PR, Brazil. Electronic address: vivian.moure@ufpr.br. [9]
DOI 10.1016/j.abb.2026.110761
PMID 41672190
发布时间 2026-07-07
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Archives of biochemistry and biophysics

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