7-Chloro-3-methyl-3-4-dihydro-2H-1,2,4 benzothiadiazine S,S-dioxide (IDRA 21): a benzothiadiazine derivative that enhances cognition by attenuating DL-alpha-amino-2,3-dihydro-5-methyl-3-oxo-4-isoxazolepropanoic acid (AMPA) receptor desensitization.
作者:
主题词
阿普唑仑(Alprazolam);动物(Animals);回避学习(Avoidance Learning);苯噻二嗪(Benzothiadiazines);脑(Brain);氯噻嗪(Chlorothiazide);认知(Cognition);二氮嗪(Diazoxide);电生理学(Electrophysiology);谷氨酸盐类(Glutamates);配体(Ligands);男(雄)性(Male);迷宫学习(Maze Learning);磷脂酰肌醇类(Phosphatidylinositols);喹恶啉类(Quinoxalines);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);受体, AMPA(Receptors, AMPA);受体, 毒蕈碱(Receptors, Muscarinic);氢溴酸东莨菪碱(Scopolamine Hydrobromide);立体异构现象(Stereoisomerism);突触体(Synaptosomes)
PMID
7815345
发布时间
2018-11-30
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