1,3-Diacylaminopropan-2-ols and corresponding 2-acyl derivatives as drug carriers: unexpected pharmacological properties.
第一作者:
D M,Lambert
第一单位:
School of Pharmacy, Laboratory of Medicinal Chemistry, Catholic University of Louvain, Brussels, Belgium.
作者:
主题词
动物(Animals);结合, 竞争性(Binding, Competitive);大脑皮质(Cerebral Cortex);药物载体(Drug Carriers);电刺激(Electric Stimulation);豚鼠(Guinea Pigs);组胺(Histamine);回肠(Ileum);肌收缩(Muscle Contraction);肌, 平滑(Muscle, Smooth);拟副交感神经药(Parasympathomimetics);丙醇胺类(Propanolamines);放射配体测定(Radioligand Assay);大鼠(Rats);受体, 阿片样, δ(Receptors, Opioid, delta);受体, 阿片样, μ(Receptors, Opioid, mu);受体, Σ(Receptors, sigma);构效关系(Structure-Activity Relationship)
DOI
10.1111/j.2042-7158.1993.tb05530.x
PMID
8097776
发布时间
2019-07-10
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