Identification of a Potent, Selective, and Efficacious Phosphatidylinositol 3-Kinase delta (P13K delta) Inhibitor for the Treatment of Immunological Disorders
第一作者:
Liu, Qingjie
作者:
Liu, Qingjie [1]
;
Shi, Qing [1]
;
Marcoux, David [1]
;
Batt, Douglas G. [1]
;
Cornelius, Lyndon [1]
;
Qin, Lan-Ying [1]
;
Ruan, Zheming [1]
;
Neels, James [1]
;
Beaudoin-Bertrand, Myra [1]
;
Srivastava, Anurag S. [1]
;
Li, Ling [1]
;
Cherney, Robert J. [2]
;
Gong, Hua [1]
;
Watterson, Scott H. [1]
;
Weigelt, Carolyn [1]
;
Gillooly, Kathleen M. [1]
;
McIntyre, Kim W. [3]
;
Xie, Jenny H. [3]
;
Obermeier, Mary T. [1]
;
Fura, Aberra [1]
;
Sleczka, Bogdan [1]
;
Stefanski, Kevin [1]
;
Fancher, R. M. [3]
;
Padmanabhan, Shweta [1]
;
Thatipamula, R. P. [1]
;
Kundu, Ipsit [1]
;
Rajareddy, Kallem [4]
;
Smith, Rodney [1]
;
Herman, James K. [1]
;
Xing, Dezhi [1]
;
Fan, Jingsong [1]
;
Levesque, Paul C. [1]
;
Ruan, Qian [3]
;
Pitt, Sidney [1]
;
Zhang, Rosemary [1]
;
Pedicord, Donna [1]
;
Pan, Jie [1]
;
Yarde, Melissa [3]
;
Lu, Hao [1]
;
Lippy, Jonathan [1]
;
Goldstine, Christine [1]
;
Skala, Stacey [1]
;
Rampulla, Richard A. [1]
;
Mathur, Arvind [1]
;
Gupta, Anuradha [1]
;
Arunachalam, Pirama Nayagam [1]
;
Sack, John S. [1]
;
Muckelbauer, Jodi K. [1]
;
Cvijic, Mary Ellen [1]
;
Salter-Cid, Luisa M. [3]
;
Bhide, Rajeev S. [1]
;
Poss, Michael A. [1]
;
Hynes, John [1]
;
Carter, Percy H. [1]
;
Macor, John E. [1]
;
Ruepp, Stefan [1]
;
Schieven, Gary L. [1]
;
Tino, Joseph A. [1]
作者单位:
Bristol Myers Squibb Co, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA
[1]
Texas Tech Univ, Hlth Sci Ctr, Sch Pharm, Amarillo, TX 79106 USA
[2]
Biocon Bristol Myers Squibb Res Ctr, Dept Discovery Synth, Biocon Pk,Bommasandra 4 Phase,Jigani Link Rd, Bengaluru 560099, India
[3]
Sanofi, Integrated Drug Discovery, 153 2nd Ave, Waltham, MA 02451 USA
[4]
发布时间
2017-12-07
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Journal of Medicinal Chemistry
Journal of Medicinal Chemistry
5193-5208页
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