Discovery of a Potent (4<i>R</i>,5<i>S</i>)-4-Fluoro-5-methylproline Sulfonamide Transient Receptor Potential Ankyrin 1 Antagonist and Its Methylene Phosphate Prodrug Guided by Molecular Modeling

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作者： Huifen Chen ^[1] ; Matthew Volgraf ^[2] ; Steven Do ^[3] ; Aleksandr Kolesnikov ^[4] ; Daniel G. Shore ; Vishal A. Verma ; Elisia Villemure ; Lan Wang ; Yong Chen ; Baihua Hu ; Ai-Jun Lu ; Guosheng Wu ; Xiaofeng Xu ; Po-wai Yuen ; Yamin Zhang ; Shawn D. Erickson ; Martin Dahl ; Christine Brotherton-Pleiss ; Suzanne Tay ; Justin Q. Ly ; Lesley J. Murray ; Jun Chen ; Desiree Amm ; Wienke Lange ; David H. Hackos ; Rebecca M. Reese ; Shannon D. Shields ; Joseph P. Lyssikatos ; Brian S. Safina ; Anthony A. Estrada

作者单位： Department of Discovery Chemistry, Department of Neurosciences, Department of Biochemical and Cellular Pharmacology, and Department of Drug Metabolism and Pharmacokinetics, Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States ^[1] Ion Channels Group, Evotec AG, Manfred Eigen Campus, Essener Bogen 7, 22419 Hamburg, Germany ^[2] Small Molecule Research, Pharmaceutical Research and Early Drug Development, Hoffmann-La Roche Inc., 340 Kingsland Street, Nutley, New Jersey 07110, United States ^[3] Pharmaron-Beijing Co. Ltd., 6 Taihe Road, BDA, Beijing 100176, P. R. China ^[4]

发布时间 2018-09-13

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Journal of Medicinal Chemistry

2018年61卷8期

3641-3659页

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Discovery of a Potent (4<i>R</i>,5<i>S</i>)-4-Fluoro-5-methylproline Sulfonamide Transient Receptor Potential Ankyrin 1 Antagonist and Its Methylene Phosphate Prodrug Guided by Molecular Modeling

Journal of Medicinal Chemistry

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Discovery of a Potent (4<i>R</i>,5<i>S</i>)-4-Fluoro-5-methylproline Sulfonamide Transient Receptor Potential Ankyrin 1 Antagonist and Its Methylene Phosphate Prodrug Guided by Molecular Modeling

Journal of Medicinal Chemistry

相似文献

Journal of Medicinal Chemistry

相关期刊

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