Discovery of a Potent Acyclic, Tripeptidic, Acyl Sulfonamide Inhibitor of Hepatitis C Virus NS3 Protease as a Back-up to Asunaprevir with the Potential for Once-Daily Dosing
第一作者:
Sun, Li-Qiang
作者:
Sun, Li-Qiang [1]
;
Mull, Eric [2]
;
Zheng, Barbara [3]
;
D'Andrea, Stanley [4]
;
Zhao, Qian [1]
;
Wang, Alan Xiangdong [1]
;
Sin, Ny [3]
;
Venables, Brian L. [5]
;
Sit, Sing-Yuen [1]
;
Chen, Yan [4]
;
Chen, Jie [6]
;
Cocuzza, Anthony [2]
;
Bilder, Donna M. [1]
;
Mathur, Arvind [3]
;
Ranipulla, Richard [5]
;
Chen, Bang-Chi [3]
;
Palani, Theerthagiri [4]
;
Ganesan, Sivakumar [4]
;
Arunachalam, Pirama Nayagam [3]
;
Falk, Paul [5]
;
Levine, Steven [7]
;
Chen, Chaoqun [8]
;
Friborg, Jacques [5]
;
Yu, Fei [5]
;
Hernandez, Dennis [8]
;
Sheaffer, Amy K. [3]
;
Knipe, Jay O. [1]
;
Han, Yong-Hae [8]
;
Schartman, Richard [5]
;
Donoso, Maria [3]
;
Mosure, Kathy [9]
;
Sinz, Michael W. [1]
;
Zvyaga, Tatyana [8]
;
Rajamani, Ramkumar [10]
;
Kish, Kevin [11]
;
Tredup, Jeffrey [3]
;
Klei, Herbert E. [3]
;
Gao, Qi [12]
;
Ng, Alicia [5]
;
Mueller, Luciano [5]
;
Grasela, Dennis M. [8]
;
Adams, Stephen [3]
;
Loy, James [3]
;
Levesaue, Paul C. [5]
;
Sun, Huabin [8]
;
Shi, Hong [13]
;
Sun, Lucy [1]
;
Warner, William [2]
;
Li, Danshi [1]
;
Zhu, Jialong [3]
;
Wang, Ying-Kai [2]
;
Fang, Hua [3]
;
Cockett, Mark I. [5]
;
Meanwell, Nicholas A. [8]
;
McPhee, Fiona [3]
;
Scola, Paul M. [3]
作者单位:
Bristol Myers Squibb Res & Dev, Dept Virol Discovery Biol, 5 Res Pkwy, Wallingford, CT 06492 USA
[1]
Bristol Myers Squibb Res & Dev, Dept Pharmaceut Dev, 1 Squibb Dr, New Brunswick, NJ 08903 USA
[2]
Bristol Myers Squibb Res & Dev, Dept Discovery Chem, 5 Res Pkwy, Wallingford, CT 06492 USA
[3]
Bristol Myers Squibb Res & Dev, Dept Lead Evaluat, 5 Res Pkwy, Wallingford, CT 06492 USA
[4]
Biocon Bristol Myers Squibb R&D Ctr, Biocon Pk,Bommasandra 4 Phase,Jigani Link Rd, Bangalore 560099, Karnataka, India
[5]
Bristol Myers Squibb Res & Dev, Dept Prot Sci & Struct, POB 5400, Princeton, NJ 08543 USA
[6]
Bristol Myers Squibb Res & Dev, Dept Clin Dev Infect Dis, POB 5400, Princeton, NJ 08543 USA
[7]
Bristol Myers Squibb Res & Dev, Dept Pharmaceut Candidate Optimizat, 5 Res Pkwy, Wallingford, CT 06492 USA
[8]
Bristol Myers Squibb Res & Dev, Dept Comp Assisted Drug Design, 5 Res Pkwy, Wallingford, CT 06492 USA
[9]
Bristol Myers Squibb Res & Dev, Dept Pharmaceut Candidate Optimizat, 311 Pennington Rocky,Hill Rd, Pennington, NJ 08534 USA
[10]
Bristol Myers Squibb Res & Dev, Dept Discovery Synth, Route 206 & Provinceline Rd, Princeton, NJ 08543 USA
[11]
Bristol Myers Squibb Res & Dev, Dept Mechanist Biochem, POB 5400, Princeton, NJ 08543 USA
[12]
Bristol Myers Squibb Res & Dev, Dept Lead Discovery & Optimizat, 5 Res Pkwy, Wallingford, CT 06492 USA
[13]
发布时间
2017-04-06
- 浏览4
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry
8042-8060页
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