首页>Bioorganic and Medicinal Chemistry Letters>Discovery and optimization of a novel CNS penetrant series of mGlu(4) PAMs based on a 1,4-thiazepane core with in vivo efficacy in a preclinical Parkinsonian model
Discovery and optimization of a novel CNS penetrant series of mGlu(4) PAMs based on a 1,4-thiazepane core with in vivo efficacy in a preclinical Parkinsonian model