Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone CBP/EP300 Bromodomain Inhibitor (CPI-637)
作者:
Taylor, Alexander M. [1]
;
Cote, Alexandre [1]
;
Hewitt, Michael C. [1]
;
Pastor, Richard [2]
;
Leblanc, Yves [2]
;
Nasveschuk, Christopher G. [3]
;
Romero, F. Anthony [1]
;
Crawford, Terry D. [1]
;
Cantone, Nico [2]
;
Jayaram, Hariharan [3]
;
Setser, Jeremy [2]
;
Murray, Jeremy [2]
;
Beresini, Maureen H. [1]
;
Boenig, Gladys de Leon [1]
;
Chen, Zhongguo [1]
;
Conery, Andrew R. [2]
;
Cummings, Richard T. [1]
;
Dakin, Leslie A. [1]
;
Flynn, E. Megan [2]
;
Huang, Oscar W. [2]
;
Kaufman, Susan [1]
;
Keller, Patricia J. [3]
;
Kiefer, James R. [3]
;
Lai, Tommy [2]
;
Li, Yingjie [3]
;
Liao, Jiangpeng [1]
;
Liu, Wenfeng [3]
;
Lu, Henry [3]
;
Pardo, Eneida [2]
;
Tsui, Vickie [2]
;
Wang, Jian [1]
;
Wang, Yongyun [3]
;
Xu, Zhaowu [2]
;
Yan, Fen [1]
;
Yu, Dong [3]
;
Zawadzke, Laura [1]
;
Zhu, Xiaoqin [1]
;
Zhu, Xiaoyu [3]
;
Sims, Robert J., III [3]
;
Cochran, Andrea G. [3]
;
Bellon, Steve [1]
;
Audia, James E. [3]
;
Magnuson, Steven [2]
;
Albrecht, Brian K. [1]
作者单位:
Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA
[1]
Wuxi AppTec Co Ltd, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China
[2]
Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA
[3]
发布时间
2017-04-05
- 浏览5
ACS medicinal chemistry letters
ACS medicinal chemistry letters
531-536页
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