新起之秀,Birabresib(OTX015/MK-8628)通过抑制BET蛋白靶向治疗NUT癌等晚期实体瘤
A Rising Star,Birabresib(MK-8628)Targets Advanced Solid Tumors Including NUT Carcinoma by Inhibiting Bromodomain and Extraterminal Proteins
摘要1 文献来源LEWIN J,SORIA J C,STATHIS A,et al.PhaseⅠb trial with birabresib,a small-molecule inhibitor of bromodomain and extraterminal proteins,in patients with selected advanced solid tumors[J].J Clin Oncol,2018,36(30):3007-3014.doi:10.1200/JCO.2018.78.2292.
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