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Pharmacokinetics,efficacy,and safety of a novel aripiprazole microsphere-based long-acting injectable formulation for schizophrenia:A multicenter,randomized controlled trial

摘要Schizophrenia is a severe and chronic psychiatric disorder with a lifetime prevalence of approximately 0.7%-1%worldwide[1].Ari-piprazole is widely used for schizophrenia treatment,and known as a dopamine system stabilizer due to its partial agonist activity as the dopamine-2(D2)and serotonin 5-hydroxytryptamine 1A(5-HT1A)receptors,as well as antagonist action at the 5-HT2A receptors[2].

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作者单位 National Clinical Research Center for Mental Disorders & National Center for Mental Disorders Beijing Anding Hospital Affiliated to Capital Medical University,Beijing,100088,China [1] Early Intervention Department,The Fourth People's Hospital of Hefei,Hefei,230022,China [2] Drug Clinical Trial Institution,The Brain Hospital Affiliated to Guangzhou Medical University,Guangzhou,510370,China [3] Medical Affairs Department,The Brain Hospital Affiliated to Guangzhou Medical University,Guangzhou,510370,China [4] Women's Psychopsychology Department,Xi'an Mental Health Center,Xi'an,710061,China [5] Psychiatric Department 6,Shandong Daizhuang Hospital,Jining,Shandong,272000,China [6] Jiangxi Provincial Psychiatric Hospital,Nanchang,220029,China [7] Female Acute Care Ward 3,Shenzhen Kangning Hospital,Shenzhen,Guangdong,518118,China [8] Beijing Huilongguan Hospital,Beijing,100096,China [9] Psychiatric Department 8,Tianjin Anding Hospital,Tianjin,300222,China [10] The 11th People's Hospital of Chongqing,Chongqing,400030,China [11] Psychosomatic Medicine Department,Deyang People's Hospital,Deyang,Sichuan,618000,China [12] Drug Clinical Trial Institution,Deyang People's Hospital,Deyang,Sichuan,618000,China [13] Premium Psychiatric Services Department,The Third People's Hospital of Huzhou,Huzhou,Zhejiang,313000,China [14] Zhuhai Livzon Microsphere Technology Co.,Ltd.,Livzon Pharmaceutical Group Inc.,Zhuhai,Guangdong,519090,China [15] Institute of Clinical Pharmacology,Peking University First Hospital,Beijing,100191,China [16]
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DOI 10.1016/j.jpha.2025.101350
发布时间 2026-06-18(万方平台首次上网日期,不代表论文的发表时间)
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药物分析学报(英文版)

药物分析学报(英文版)

2026年16卷1期

305-308页

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